SCHEMBL21887582

SCHEMBL21887582

C=C1/C(=C\C=C/C)C2(c3ccccc3-c3ccccc32)c2ccc3oc4ccc(-c5ccc(-c6nc7ccccc7n6-c6ccccc6)cc5)cc4c3c21

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
PRKACA P17612 1/20 0.30
RPS6KB1 P23443 1/20 0.30
GSK3B P49841 1/20 0.30
ROCK1 Q13464 1/20 0.30
GRIA1 P42261 1/20 0.30
CACNG8 Q8WXS5 1/20 0.30
CACNG2 Q9Y698 1/20 0.30
PTGER4 P35408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18156764 0.84 ESR1 (0.39) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL22423178 0.83 PTGER4 (0.30) PTGER4
SCHEMBL18156765 0.78 ESR1 (0.37) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL18156731 0.76 ESR1 (0.38) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL20224492 0.76 RECQL (0.36) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL18156738 0.74 ESR1 (0.42) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL20224493 0.73 SIRT2 (0.33) ESR1ESR2PTGER4
SCHEMBL18156735 0.73 RECQL (0.38) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL18156732 0.72 ESR1 (0.39) RECQLESR1ESR2PRKACARPS6KB1
SCHEMBL20248537 0.72 RECQL (0.35) RECQLESR1ESR2PRKACARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3083880-B1 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2020-04-01 EP disclosed