SCHEMBL2189564

SCHEMBL2189564

CC(C)c1ccc(CC(=O)NCc2nc(C(=O)NCCc3ccccc3F)cs2)cc1.NC(=O)c1nc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)sc1Cc1c(F)cccc1F.NC(=O)c1nc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)sc1Cc1cccc(F)c1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.35
IGF1R P08069 1/20 0.33
ALDH1A1 P00352 1/20 0.33
THRB P10828 1/20 0.32
MAPT P10636 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LTA4H P09960 1/20 0.31
EPHX2 P34913 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNA1H O95180 1/20 0.31
CNR2 P34972 1/20 0.31
KCNH2 Q12809 1/20 0.31
CACNA1I Q9P0X4 1/20 0.31
TP53 P04637 2/20 0.31
PREP P48147 1/20 0.31
FAP Q12884 1/20 0.31
SLC40A1 Q9NP59 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2189562 0.88 TRPV1 (0.40) TRPV1IGF1RALDH1A1THRBMAPT
SCHEMBL5668846 0.79 IGF1R (0.47) IGF1RMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL2172634 0.78 TRPV1 (0.56) TRPV1IGF1RMAPTCYP1A2CYP3A4
SCHEMBL2189359 0.74 CNR1 (0.33) TRPV1ALDH1A1MAPTTP53
SCHEMBL2175901 0.72 SCN2A (0.47) TRPV1IGF1RMAPTCYP1A2CYP3A4
SCHEMBL2186614 0.71 TRPV1 (0.40) TRPV1IGF1RMAPTCYP1A2CYP3A4
SCHEMBL4387635 0.70 SGMS1 (0.47) TRPV1ALDH1A1THRBMAPTCYP1A2
SCHEMBL2172869 0.70 CYP1A2 (0.43) TRPV1ALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL4390454 0.70 MAPT (0.46) TRPV1ALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL4392420 0.70 CYP1A2 (0.52) ALDH1A1MAPTCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed