SCHEMBL21901422

SCHEMBL21901422

C=CC(=O)N1CCN(c2ncnc3c(C)c(-c4cc(O)cc5ccccc45)c(Cl)cc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.61
EGFR P00533 1/20 0.56
HMOX2 P30519 1/20 0.56
CRYZ Q08257 1/20 0.56
VAT1 Q99536 1/20 0.56
RTN4 Q9NQC3 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29715195 0.90 KRAS (0.72) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647122 0.90 KRAS (0.72) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765855 0.89 KRAS (0.58) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647214 0.89 KRAS (0.58) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647072 0.83 KRAS (0.60) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765992 0.83 KRAS (0.60) KRASEGFRHMOX2CRYZVAT1
SCHEMBL17026609 0.83 KRAS (0.60) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647142 0.82 KRAS (0.72) KRAS
SCHEMBL29765748 0.82 KRAS (0.72) KRAS
SCHEMBL18134007 0.82 KRAS (0.70) KRASEGFRHMOX2CRYZVAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081282-A1 KRAS G12C INHIBITORS ELI LILLY AND COMPANY (US) 2020-04-23 WO disclosed