SCHEMBL21936052

SCHEMBL21936052

CC(C)C(=O)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.48
LIPG Q9Y5X9 6/20 0.43
LPL P06858 5/20 0.43
F11 P03951 3/20 0.39
F2 P00734 2/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
P4HB P07237 1/20 0.36
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA9 Q16790 4/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
AAK1 Q2M2I8 2/20 0.35
CA12 O43570 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3502436 0.89 ROCK1 (0.46) ROCK1LIPGLPLF11F2
SCHEMBL794033 0.84 ROCK1 (0.48) ROCK1LIPGLPLF11F2
SCHEMBL1130871 0.84 ROCK1 (0.48) ROCK1LIPGLPLF11F2
SCHEMBL16035253 0.82 ROCK1 (0.47) ROCK1LIPGLPLF11F2
SCHEMBL1044923 0.82 ROCK1 (0.47) ROCK1LIPGLPLF11F2
SCHEMBL15594472 0.80 ROCK1 (0.46) ROCK1LIPGLPLF11F2
SCHEMBL793338 0.80 ROCK1 (0.48) ROCK1LIPGLPLF11F2
SCHEMBL12069299 0.80 ROCK1 (0.46) ROCK1LIPGLPLF11F2
SCHEMBL516413 0.80 ROCK1 (0.46) ROCK1LIPGLPLF11F2
SCHEMBL28960278 0.80 ROCK1 (0.46) ROCK1LIPGLPLF11F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
CN-112601745-A Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2021-04-02 CN disclosed
WO-2020082921-A1 NITROGEN HETEROARYL AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2020-04-30 WO disclosed