SCHEMBL21953141

SCHEMBL21953141

Cc1nc(Nc2ccc(C=N)c(N)c2)cc(-c2cc(Cl)ccc2C)n1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 17/20 0.57
TP53 P04637 2/20 0.46
MAPT P10636 2/20 0.46
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21953110 0.89 AGPAT2 (0.59) AGPAT2TP53MAPT
SCHEMBL4288850 0.80 AGPAT2 (0.74) AGPAT2TP53MAPTNPC1CYP1A2
SCHEMBL4279343 0.76 AGPAT2 (0.77) AGPAT2TP53MAPTLMNAPOLB
SCHEMBL13880171 0.73 AGPAT2 (1.00) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL25039650 0.73 AGPAT2 (0.53) AGPAT2TP53MAPTLMNAPOLB
SCHEMBL4287579 0.72 AGPAT2 (0.62) AGPAT2TP53MAPTNPC1RAB9A
SCHEMBL13880169 0.71 AGPAT2 (0.90) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL13880176 0.69 AGPAT2 (1.00) AGPAT2MAPTNPC1CYP1A2CYP3A4
SCHEMBL13880262 0.69 AGPAT2 (0.88) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL13892055 0.68 AGPAT2 (0.77) AGPAT2NPC1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO disclosed