SCHEMBL2196884

SCHEMBL2196884

O=S(=O)(c1ccc(C(OC2CCCC2)c2nc3nccnc3[nH]2)cc1)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 1/20 0.40
GCK P35557 14/20 0.39
LNPEP Q9UIQ6 1/20 0.36
CDK1 P06493 3/20 0.34
CDK2 P24941 3/20 0.34
KDR P35968 3/20 0.34
CDK4 P11802 1/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2177869 0.79 GCK (0.44) PIK3C3GCKLNPEP
SCHEMBL2198311 0.78 GCK (0.60) PIK3C3GCKLNPEP
SCHEMBL2180026 0.71 GCK (0.48) GCK
SCHEMBL2196374 0.70 GCK (0.51) GCKNAMPT
SCHEMBL2177573 0.68 GCK (0.43) GCKNAMPT
SCHEMBL2280345 0.68 GCK (0.47) GCKNAMPT
SCHEMBL2280341 0.68 GCK (0.47) GCKNAMPT
SCHEMBL2180158 0.67 GCK (0.46) GCK
SCHEMBL2198514 0.67 GCK (0.50) GCKNAMPT
SCHEMBL2415677 0.67 CDK1 (0.34) GCKLNPEPCDK1CDK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO disclosed