SCHEMBL21976503

SCHEMBL21976503

CSc1ccc(C2Nc3ccc(C(=O)NO)cc3N2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
GAA P10253 2/20 0.45
KMT2A Q03164 2/20 0.45
NPC1 O15118 1/20 0.45
PLK1 P53350 1/20 0.42
HDAC1 Q13547 6/20 0.40
HDAC6 Q9UBN7 6/20 0.40
HDAC8 Q9BY41 4/20 0.40
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALOX5 P09917 1/20 0.36
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
BLM P54132 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21975936 0.96 MEN1 (0.42) MEN1GAAKMT2ANPC1PLK1
SCHEMBL21976310 0.81 HDAC6 (0.37) MEN1GAAKMT2APLK1HDAC1
SCHEMBL23677092 0.78 HDAC6 (0.42) PLK1HDAC1HDAC6HDAC8POLB
SCHEMBL21976470 0.76 HDAC6 (0.55) MEN1KMT2ANPC1HDAC1HDAC6
SCHEMBL21976251 0.76 HDAC6 (0.52) HDAC1HDAC6HDAC8HDAC3HDAC4
SCHEMBL21975922 0.75 MEN1 (0.53) MEN1GAAKMT2ANPC1HDAC6
SCHEMBL21976950 0.75 HDAC1 (0.47) GAAHDAC1HDAC6HDAC8KDM4E
SCHEMBL21976968 0.75 HDAC6 (0.50) HDAC1HDAC6HDAC8ALOX5HDAC3
SCHEMBL13485782 0.74 PLK1 (0.70) NPC1PLK1HDAC1HDAC6HDAC8
SCHEMBL21976291 0.74 KDM1A (0.43) MEN1KMT2ANPC1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed