SCHEMBL21986390

SCHEMBL21986390

COCCN1C[C@@H]2C(I)[C@@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.44
HSD11B1 P28845 1/20 0.33
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32
KDM1A O60341 1/20 0.32
MAP3K12 Q12852 7/20 0.32
KAT2B Q92831 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814858 0.80 GBA1 (0.46) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL20115401 0.80 GBA1 (0.46) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL24461156 0.77 GBA1 (0.43) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL22098589 0.75 GBA1 (0.42) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL26790067 0.75 GBA1 (0.42) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL20115395 0.75 GBA1 (0.42) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL18484868 0.75
SCHEMBL19938007 0.75 GBA1 (0.48) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL23851396 0.74 GBA1 (0.41) GBA1HSD11B1CYP2D6SLC6A2SLC6A4
SCHEMBL23851395 0.74 GBA1 (0.41) GBA1HSD11B1CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3172214-B1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2020-05-13 EP disclosed