SCHEMBL21990149

SCHEMBL21990149

Cc1ccc(CNC(=O)c2ccc3c(c2)N(Cc2ccc(F)c(F)c2)C(=O)C3(C)C)o1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 2/20 0.50
TP53 P04637 2/20 0.43
HTR7 P34969 1/20 0.41
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40
CPT1B Q92523 1/20 0.40
PPARG P37231 1/20 0.39
SCN9A Q15858 1/20 0.38
MAPT P10636 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1I Q9P0X4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21990157 0.91 STING1 (0.54) STING1TP53CPT2CPT1ACPT1B
SCHEMBL21990102 0.89 STING1 (0.56) STING1TP53HTR7CPT2CPT1A
SCHEMBL21990122 0.86 STING1 (0.64) STING1TP53CPT2CPT1ACPT1B
SCHEMBL21990167 0.86 STING1 (0.52) STING1TP53MAPT
SCHEMBL20594920 0.85 TP53 (0.38) STING1TP53HTR7PPARGSCN9A
SCHEMBL21989990 0.85 STING1 (0.44) STING1TP53CPT2CPT1ACPT1B
SCHEMBL21990173 0.84 STING1 (0.55) STING1TP53CPT2CPT1ACPT1B
SCHEMBL21990031 0.84 STING1 (0.61) STING1TP53CPT2CPT1ACPT1B
SCHEMBL21990069 0.84 STING1 (0.54) STING1TP53HTR7CPT2CPT1A
SCHEMBL21990068 0.83 STING1 (0.74) STING1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200172483-A1 HETEROCYCLIC SMALL MOLECULE MODULATORS OF HUMAN STING CURADEV PHARMA LIMITED (GB) 2020-06-04 US claimed
US-20200172483-A1 HETEROCYCLIC SMALL MOLECULE MODULATORS OF HUMAN STING CURADEV PHARMA LIMITED (GB) 2020-06-04 US disclosed
US-20200172483-A1 HETEROCYCLIC SMALL MOLECULE MODULATORS OF HUMAN STING CURADEV PHARMA LIMITED (GB) 2020-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200172483-A1 HETEROCYCLIC SMALL MOLECULE MODULATORS OF HUMAN STING STING1, IRF3, CGAS STING1 1/4885TP53 131/4885HTR7 3469/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.