SCHEMBL21994243

SCHEMBL21994243

O=C(Cc1ccccc1)NC1CNCC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.74
CYP3A4 P08684 3/20 0.74
CYP2D6 P10635 3/20 0.74
CYP2C19 P33261 3/20 0.74
CYP2C9 P11712 2/20 0.74
SIGMAR1 Q99720 3/20 0.50
MAOA P21397 2/20 0.50
CNR2 P34972 1/20 0.49
AKT1 P31749 1/20 0.46
MC4R P32245 1/20 0.45
LTA4H P09960 1/20 0.44
EPHX2 P34913 1/20 0.44
KDM1A O60341 1/20 0.43
MAOB P27338 1/20 0.43
MAPK1 P28482 1/20 0.42
P2RX7 Q99572 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994288 0.88 KCNH2 (0.75) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994284 0.88 KCNH2 (0.78) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994242 0.87 KCNH2 (0.67) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994254 0.85 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994239 0.85 KCNH2 (1.00) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994246 0.85 KCNH2 (0.74) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994259 0.84 KCNH2 (0.63) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994286 0.82 KCNH2 (0.68) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL22053368 0.81 KCNH2 (0.79) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL21994241 0.78 KCNH2 (1.00) KCNH2CYP3A4CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020107189-A1 PYRROLIDINE COMPOUNDS FOR THE TREATMENT OF MALARIA LEGION PHARMA CO. LTD (CN) 2020-06-04 WO claimed