SCHEMBL21996499

SCHEMBL21996499

COC1CCN(C(=O)OC(C)(C)C)C12CC2(Br)Br

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.33
RECQL P46063 1/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX1 P07099 1/20 0.33
PREP P48147 2/20 0.32
ALDH1A1 P00352 1/20 0.32
EPHX2 P34913 1/20 0.32
GPR119 Q8TDV5 2/20 0.32
KDM1A O60341 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21996530 0.81 CHRM2 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL21996585 0.77 KLK7 (0.43) SMN1; SMN2GPR119DDB1CRBNKDM4E
SCHEMBL21996435 0.77 CHRM2 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL24622087 0.77 CHRM2 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL28762092 0.77 CHRM2 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL28735702 0.75 HSD17B10 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL29519627 0.75 HSD17B10 (0.36) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL25349844 0.70 MEN1 (0.34) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL25348114 0.70 MEN1 (0.34) CHRM2CHRM1CHRM3HPGDHSD17B10
SCHEMBL30782508 0.70 MEN1 (0.34) CHRM2CHRM1CHRM3HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113077-A9 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-08-13 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed