SCHEMBL2200537

SCHEMBL2200537

CCC1C(CC(=O)O)CCCN1c1c(F)cc2c(=O)c(C(=O)NCc3ccc(Cl)cc3Cl)cn(CC(F)(F)F)c2c1OC

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 9/20 0.41
SMN1; SMN2 Q16637 1/20 0.36
P2RX7 Q99572 2/20 0.35
PDE10A Q9Y233 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2199871 0.86 TOP1 (0.51) TOP1P2RX7POLB
SCHEMBL2202775 0.83 TOP1 (0.49) TOP1P2RX7
SCHEMBL1974822 0.82 TOP1 (0.48) TOP1P2RX7POLB
SCHEMBL12427312 0.81 TOP1 (0.47) TOP1P2RX7POLB
SCHEMBL12427350 0.81 TOP1 (0.48) TOP1P2RX7
SCHEMBL2207572 0.81 TOP1 (0.46) TOP1SMN1; SMN2
SCHEMBL13744618 0.80 TOP1 (0.45) TOP1P2RX7POLB
SCHEMBL4251735 0.80 TOP1 (0.45) TOP1P2RX7POLB
SCHEMBL13744928 0.80 TOP1 (0.45) TOP1P2RX7POLB
SCHEMBL1971493 0.80 TOP1 (0.45) TOP1P2RX7PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977349-B2 Substituted quinolones III AICURIS GMBH & CO. KG (DE) 2011-07-12 US disclosed