SCHEMBL22006155

SCHEMBL22006155

O=C(N1Cc2cccnc2Nc2ccccc21)C12CC3C1C32

nearest known ligand 0.72

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 20/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27486147 0.84 IDH1 (0.73) IDH1
SCHEMBL17807045 0.84 IDH1 (1.00) IDH1
SCHEMBL19713523 0.82 IDH1 (1.00) IDH1
SCHEMBL19725577 0.82 IDH1 (1.00) IDH1
SCHEMBL19713522 0.82 IDH1 (1.00) IDH1
SCHEMBL17806802 0.80 IDH1 (1.00) IDH1
SCHEMBL17806760 0.80 IDH1 (0.80) IDH1
SCHEMBL22006165 0.80 IDH1 (0.70) IDH1
SCHEMBL17806729 0.79 IDH1 (1.00) IDH1
SCHEMBL19713551 0.78 IDH1 (1.00) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3226690-B1 NOVEL TRICYCLIC COMPOUNDS AS INHIBITORS OF MUTANT IDH ENZYMES MERCK SHARP & DOHME (US) 2020-05-20 EP disclosed