SCHEMBL2200918

SCHEMBL2200918

Cc1nn(-c2cccc(OC(F)(F)F)c2)c(C2CC2)c1C(=O)N1CCC(N2C[C@@H](O)C[C@H]2C)CC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
SCN9A Q15858 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
NOTUM Q6P988 1/20 0.38
HSD11B1 P28845 1/20 0.37
MGLL Q99685 1/20 0.37
MAPK7 Q13164 4/20 0.36
MAPT P10636 1/20 0.36
CCKAR P32238 1/20 0.36
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
OPRM1 P35372 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CSNK1E P49674 1/20 0.35
TP53 P04637 1/20 0.35
CCR5 P51681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2202132 1.00 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2198057 1.00 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2200049 1.00 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2201212 0.88 HRH3 (0.41) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL13973649 0.88 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2201691 0.88 SCN9A (0.41) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL12429708 0.87 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2203329 0.87 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL12429781 0.87 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1
SCHEMBL2203789 0.87 KMT2A (0.40) KMT2ASCN9ASCN10ANOTUMHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977358-B2 Pyrazol derivatives HOFFMANN-LA ROCHE INC. (US) 2011-07-12 US disclosed