SCHEMBL22013132

SCHEMBL22013132

OC1CCN(SNc2ccnc3ccc(N4CCC(F)C4)nc23)C1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 9/20 0.39
MELK Q14680 1/20 0.36
PDE10A Q9Y233 2/20 0.36
P2RX7 Q99572 4/20 0.35
BRAF P15056 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23837023 0.80 MKNK1 (0.41) MAP4K4MELKPDE10AP2RX7
SCHEMBL22013239 0.80 MKNK1 (0.41) MAP4K4MELKPDE10AP2RX7
SCHEMBL22013104 0.79 MELK (0.39) MAP4K4MELKPDE10AP2RX7BRAF
SCHEMBL23836947 0.79 MELK (0.39) MAP4K4MELKPDE10AP2RX7BRAF
SCHEMBL23837000 0.79 MELK (0.38) MAP4K4MELKPDE10AP2RX7BRAF
SCHEMBL23836944 0.75 MAP4K4 (0.52) MAP4K4PDE10A
SCHEMBL23837065 0.74 MAP4K4 (0.37) MAP4K4MELKPDE10AP2RX7BRAF
SCHEMBL23836964 0.74 MAP4K4 (0.37) MAP4K4MELKPDE10AP2RX7BRAF
SCHEMBL23836955 0.72 MAP4K4 (0.53) MAP4K4PDE10A
SCHEMBL23837028 0.72 MAP4K4 (0.47) MAP4K4PDE10AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed