SCHEMBL22013651

SCHEMBL22013651

O=C(Nc1ccnc2ccc(N3CCCC3)nc12)c1cnc(N2CC[C@H](O)C2)nc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.41
HDAC6 Q9UBN7 2/20 0.40
MELK Q14680 2/20 0.40
MCHR1 Q99705 1/20 0.39
DGAT1 O75907 1/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HPGDS O60760 1/20 0.37
HDAC1 Q13547 2/20 0.37
PDE10A Q9Y233 1/20 0.37
DGAT2 Q96PD7 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
GSK3B P49841 1/20 0.36
ABL1 P00519 1/20 0.36
FASN P49327 1/20 0.36
NAPEPLD Q6IQ20 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23837038 0.90 MAPT (0.45) MAP4K4HDAC6MELKMAPTALDH1A1
SCHEMBL22013100 0.82 NTRK1 (0.51)
SCHEMBL29692846 0.82 NTRK1 (0.51)
SCHEMBL28596748 0.82 NTRK1 (0.51)
SCHEMBL22014119 0.81 MAP4K4 (0.41) MAP4K4MELKDGAT2
SCHEMBL23837076 0.81 MAP4K4 (0.41) MAP4K4MELKDGAT2
SCHEMBL22013375 0.76 PDE10A (0.45) MAP4K4MELKPDE10A
SCHEMBL23837016 0.76 PDE10A (0.45) MAP4K4MELKPDE10A
SCHEMBL22083650 0.73 NTRK1 (0.47) HDAC6IRAK4
SCHEMBL23836947 0.73 MELK (0.39) MAP4K4MELKPDE10ADGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed