SCHEMBL22014308

SCHEMBL22014308

O=P(O)(O)CN1CCN(CP(=O)(O)c2ccccc2)CCN(CP(=O)(O)c2ccc(P(=O)(O)CN3CCNCCNCC3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.41
SIGMAR1 Q99720 4/20 0.41
MAPT P10636 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN4 P29074 1/20 0.34
PTPN9 P43378 1/20 0.34
PTPN11 Q06124 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22014482 0.88 CFTR (0.52) CFTRALDH1A1MEN1KMT2APTPN2
SCHEMBL22014092 0.88 CFTR (0.52) CFTRALDH1A1MEN1KMT2APTPN2
SCHEMBL22014317 0.83 CFTR (0.57) CFTRALDH1A1MEN1KMT2APTPN2
SCHEMBL8393831 0.78 MAPT (0.49) SIGMAR1MAPTCHRM2CHRM5CHRM1
SCHEMBL9041381 0.78 MAPT (0.49) SIGMAR1MAPTCHRM2CHRM5CHRM1
SCHEMBL336114 0.78 MAPT (0.49) SIGMAR1MAPTCHRM5CHRM3ALDH1A1
SCHEMBL472195 0.78 MAPT (0.49) SIGMAR1MAPTCHRM5CHRM3ALDH1A1
SCHEMBL336756 0.76 MAPT (0.50) SIGMAR1MAPTCHRM5CHRM3MEN1
SCHEMBL7453394 0.76 MAPT (0.50) SIGMAR1MAPTCHRM5CHRM3MEN1
SCHEMBL21961918 0.76 CFTR (0.48) CFTRALDH1A1MEN1KMT2APTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102820-A1 COMPOUNDS FOR USE AS IRON (III) MRI CONTRAST AGENTS CONTAINING ANIONIC PENDENTS AND ANCILLARY GROUPS THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-05-22 WO disclosed