SCHEMBL22061369

SCHEMBL22061369

Cc1nn2c(=O)c(Br)cc(Cl)c2c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 6/20 0.38
CDK4 P11802 6/20 0.35
CCND1 P24385 6/20 0.35
CCNE2 O96020 2/20 0.32
CCNE1 P24864 2/20 0.32
CDK2 P24941 2/20 0.32
HAVCR2 Q8TDQ0 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
PARP1 P09874 2/20 0.32
PTGES O14684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22060800 0.67 MKNK1 (0.48)
SCHEMBL5863360 0.65 PARP1 (0.38) PDE2ACDK4CCND1PARP1
SCHEMBL7603458 0.63 PDE2A (0.36) PDE2APARP1
SCHEMBL5863219 0.62 PDE2A (0.39) PDE2ACDK4CCND1PARP1
SCHEMBL3123895 0.62 GRIN2D (0.41)
SCHEMBL11396433 0.61 PDE2A (0.47) PDE2A
SCHEMBL18362225 0.61 PDE2A (0.39) PDE2A
SCHEMBL21957279 0.60 GRIA1 (0.34)
SCHEMBL25112475 0.59 CDK4 (0.42) PDE2ACDK4CCND1PARP1
SCHEMBL30826923 0.59 KDM4E (0.55) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111253397-B MNK inhibitors 上海迪诺医药科技有限公司 2023-11-14 CN disclosed
CN-111253397-A MNK inhibitors 上海迪诺医药科技有限公司 2020-06-09 CN disclosed
WO-2020108619-A1 MNK INHIBITOR 上海迪诺医药科技有限公司 2020-06-04 WO disclosed