SCHEMBL22065403

SCHEMBL22065403

Cc1ccc(C(=O)Nc2cccc(N)c2)cc1NI

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
PTGS1 P23219 2/20 0.54
DDX3X O00571 2/20 0.54
BTK Q06187 10/20 0.48
BLK P51451 7/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
KCNK3 O14649 1/20 0.48
KCNH2 Q12809 1/20 0.48
KCNK9 Q9NPC2 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
LCK P06239 1/20 0.47
KIT P10721 1/20 0.47
SRC P12931 1/20 0.47
MAPK14 Q16539 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22065290 0.85 MEN1 (0.61) ALDH1A1SMN1; SMN2KDM4EMAPTKCNK3
SCHEMBL22066357 0.85 HDAC8 (0.58) MAPTKCNK3KCNK9MEN1KMT2A
SCHEMBL22025447 0.85 PTGS1 (0.55) ALDH1A1SMN1; SMN2PTGS1DDX3XBTK
SCHEMBL22065294 0.84 KCNK3 (0.58) ALDH1A1SMN1; SMN2KDM4EMAPTKCNK3
SCHEMBL22065293 0.84 MAOB (0.53) ALDH1A1SMN1; SMN2KDM4EMAPTKCNK3
SCHEMBL22065295 0.84 KCNK3 (0.58) SMN1; SMN2KCNK3KCNK9MEN1KMT2A
SCHEMBL22065405 0.82 RXFP1 (0.67) ALDH1A1SMN1; SMN2KDM4EMAPTKCNK3
SCHEMBL16430819 0.81 NPC1 (0.62) ALDH1A1SMN1; SMN2PTGS1DDX3XBTK
SCHEMBL22065302 0.81 KIT (0.71) KDM4EMAPTKCNK3KCNK9MEN1
SCHEMBL29568808 0.80 PTGS1 (0.79) ALDH1A1SMN1; SMN2PTGS1DDX3XMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed