SCHEMBL22065404

SCHEMBL22065404

CNc1cc(C(=O)Nc2cccc(OC)c2)ccc1C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.68
NPC1 O15118 8/20 0.67
RAB9A P51151 7/20 0.67
SMN1; SMN2 Q16637 4/20 0.67
ALDH1A1 P00352 3/20 0.67
TP53 P04637 2/20 0.67
KMT2A Q03164 2/20 0.67
PKM P14618 1/20 0.67
MAPT P10636 2/20 0.65
NLRP3 Q96P20 1/20 0.63
KCNK3 O14649 2/20 0.61
KCNK9 Q9NPC2 2/20 0.61
TRPV1 Q8NER1 1/20 0.61
HTT P42858 1/20 0.60
PLAU P00749 1/20 0.59
KDM4E B2RXH2 1/20 0.59
MEN1 O00255 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22065405 0.89 RXFP1 (0.67) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL22025452 0.86 RXFP1 (0.64) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL22065214 0.85 NPC1 (0.62) NPC1RAB9AALDH1A1MAPTKCNK3
SCHEMBL22065291 0.84 MEN1 (0.68) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL10055020 0.83 NPC1 (0.94) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL22025454 0.83 RXFP1 (0.70) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL4251080 0.82 NPC1 (0.81) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL30862297 0.82 RXFP1 (0.94) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL4251968 0.82 RXFP1 (0.94) RXFP1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL22065285 0.82 BRAF (0.60) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed