SCHEMBL22069747

SCHEMBL22069747

O=[N+]([O-])c1ccc(OCC2CCCC2)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.59
S1PR4 O95977 1/20 0.52
HSPB1 P04792 5/20 0.47
CNR2 P34972 1/20 0.45
SIGMAR1 Q99720 2/20 0.44
NPBWR1 P48145 1/20 0.44
MCHR1 Q99705 1/20 0.44
ALDH1A1 P00352 2/20 0.42
TLR4 O00206 1/20 0.41
TLR2 O60603 1/20 0.41
HIF1A Q16665 1/20 0.41
PARP10 Q53GL7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2551985 0.94 S1PR4 (0.54) CYP19A1S1PR4HSPB1CNR2SIGMAR1
SCHEMBL30879298 0.89 CYP19A1 (0.62) CYP19A1S1PR4HSPB1CNR2SIGMAR1
SCHEMBL13419634 0.88 S1PR4 (0.49) CYP19A1S1PR4HSPB1SIGMAR1ALDH1A1
SCHEMBL30152356 0.87 S1PR4 (0.48) CYP19A1S1PR4HSPB1SIGMAR1
SCHEMBL3213149 0.86 SCN9A (0.48) CYP19A1S1PR4HSPB1
SCHEMBL13419646 0.86 S1PR4 (0.50) CYP19A1S1PR4HSPB1SIGMAR1ALDH1A1
SCHEMBL3203873 0.85 CYP19A1 (0.48) CYP19A1S1PR4HSPB1SIGMAR1
SCHEMBL22069670 0.83 CYP19A1 (0.57) CYP19A1CNR2ALDH1A1
SCHEMBL28844678 0.83 CYP19A1 (0.55) CYP19A1S1PR4HSPB1SIGMAR1ALDH1A1
SCHEMBL5704513 0.82 CYP19A1 (0.62) CYP19A1NPBWR1MCHR1ALDH1A1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed