SCHEMBL22072085

SCHEMBL22072085

OCC1CCCN1c1nc(Nc2cc(C3CC3)[nH]n2)c2ccccc2n1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 3/20 0.66
PAK1 Q13153 3/20 0.66
NTRK1 P04629 2/20 0.55
ULK1 O75385 1/20 0.53
SRC P12931 1/20 0.52
CCNA2 P20248 1/20 0.52
CDK2 P24941 1/20 0.52
GSK3B P49841 1/20 0.52
NTRK3 Q16288 1/20 0.51
NTRK2 Q16620 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31471765 0.81 PAK4 (0.81) PAK4PAK1SRCCCNA2CDK2
SCHEMBL31471889 0.81 PAK4 (0.74) PAK4PAK1
SCHEMBL31141210 0.80 PAK4 (0.61) PAK4PAK1NTRK1ULK1SRC
SCHEMBL22072524 0.79 PAK4 (0.83) PAK4PAK1
SCHEMBL31471972 0.79 PAK4 (0.83) PAK4PAK1
SCHEMBL22072090 0.77 PAK4 (0.77) PAK4PAK1
SCHEMBL31471946 0.77 PAK4 (0.65) PAK4PAK1NTRK1ULK1SRC
SCHEMBL31472008 0.77 PAK4 (0.65) PAK4PAK1NTRK1ULK1SRC
SCHEMBL3644297 0.77 CDK1 (0.62) CDK2
SCHEMBL3644294 0.77 CDK1 (0.62) CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed