SCHEMBL2207232

SCHEMBL2207232

CCOP(=O)(OCC)C(C#N)Cc1ccc(C(=O)Nc2cc(-c3cccs3)ccc2N)cc1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.71
HDAC2 Q92769 4/20 0.67
HDAC3 O15379 1/20 0.67
HDAC8 Q9BY41 1/20 0.67
KCNH2 Q12809 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12434658 0.91 HDAC1 (0.69) HDAC1HDAC2HDAC3HDAC8
SCHEMBL2209274 0.90 HDAC1 (0.75) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL4316268 0.89 HDAC1 (0.66) HDAC1HDAC2HDAC3
SCHEMBL2210334 0.87 HDAC1 (0.69) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL2209831 0.87 HDAC1 (0.72) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL2206276 0.86 HDAC1 (0.53) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL2211204 0.84 HDAC1 (0.75) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL2212087 0.83 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC8
SCHEMBL8222152 0.83 KCNH2 (0.74) HDAC1HDAC2HDAC3HDAC8KCNH2
SCHEMBL2209245 0.83 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7981874-B2 Phosphorus derivatives as histone deacetylase inhibitors MERCK SHARP & DOHME CORP. (US) 2011-07-19 US claimed
US-7981874-B2 Phosphorus derivatives as histone deacetylase inhibitors MERCK SHARP & DOHME CORP. (US) 2011-07-19 US disclosed