SCHEMBL2209044

SCHEMBL2209044

CC(C)N1CCC(Oc2cccc3ccc(C(=O)N4CCCC4C)nc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.58
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.41
MCHR1 Q99705 6/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214389 0.94 HRH3 (0.52) HRH3ALDH1A1MCHR1HCRTR1HCRTR2
SCHEMBL2206395 0.92 HRH3 (0.48) HRH3ALDH1A1POLBMCHR1HCRTR1
SCHEMBL2208187 0.87 HRH3 (0.48) HRH3POLBMCHR1
SCHEMBL2209033 0.87 HRH3 (0.68) HRH3POLBMCHR1
SCHEMBL2210278 0.87 HRH3 (0.68) HRH3POLBMCHR1
SCHEMBL2208189 0.86 HRH3 (0.64) HRH3MCHR1
SCHEMBL2208886 0.86 HRH3 (0.61) HRH3MCHR1KMT2A
SCHEMBL2209751 0.85 HRH3 (0.53) HRH3MCHR1
SCHEMBL2211215 0.84 HRH3 (0.57) HRH3MCHR1
SCHEMBL2211838 0.83 HRH3 (0.52) HRH3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805166-B1 QUINOLINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-07-27 EP claimed