SCHEMBL22097771

SCHEMBL22097771

Cn1cc(Nc2ncc(Cl)c(-c3ccc(C(=O)O)cc3)n2)cn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK19 Q9BWU1 1/20 0.56
ALK Q9UM73 1/20 0.56
CDK2 P24941 4/20 0.55
CDK9 P50750 4/20 0.55
CCNT1 O60563 3/20 0.55
CCNB2 O95067 3/20 0.55
CCNE2 O96020 3/20 0.55
CDK1 P06493 3/20 0.55
CCNB1 P14635 3/20 0.55
CCNE1 P24864 3/20 0.55
CDK5 Q00535 3/20 0.55
CDK5R1 Q15078 3/20 0.55
CCNB3 Q8WWL7 3/20 0.55
KDR P35968 8/20 0.52
AURKB Q96GD4 6/20 0.52
JAK2 O60674 2/20 0.52
CDC7 O00311 1/20 0.52
DAPK3 O43293 1/20 0.52
ROCK2 O75116 1/20 0.52
PRKD3 O94806 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22097773 0.89 CDK2 (0.53) CDK19ALKCDK2CDK9CCNT1
SCHEMBL22097741 0.88 JAK2 (0.54) KDRAURKBJAK2GSK3BFLT4
SCHEMBL22097889 0.86 HDAC3 (0.51) CDK2CDK9CCNT1CCNB2CCNE2
SCHEMBL31557663 0.86 HDAC3 (0.51) CDK2CDK9CCNT1CCNB2CCNE2
SCHEMBL22544660 0.86 CDK19 (0.57) CDK19ALKCDK2CDK9CCNT1
SCHEMBL29754198 0.86 CDK19 (0.57) CDK19ALKCDK2CDK9CCNT1
SCHEMBL24853418 0.86 AURKA (0.50) CDK2CDK9CCNT1CCNB2CCNE2
SCHEMBL31557666 0.86 HDAC3 (0.51) CDK9KDRAURKBJAK2CDK7
SCHEMBL31557670 0.86 AURKA (0.50) CDK2CDK9CCNT1CCNB2CCNE2
SCHEMBL22097934 0.86 HDAC3 (0.51) CDK9KDRAURKBJAK2CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250115586-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO LTD (CN) 2025-04-10 US disclosed
US-12030870-B2 Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof LYNK PHARMACEUTICALS CO. LTD. (CN) 2024-07-09 US disclosed
US-12030870-B2 Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof LYNK PHARMACEUTICALS CO. LTD. (CN) 2024-07-09 US disclosed
US-20240025882-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2024-01-25 US disclosed
US-20240025882-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2024-01-25 US disclosed
US-20230002362-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2023-01-05 US disclosed
WO-2020119819-A1 BENZAMIDES OF PYRAZOLYL-AMINO-PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2020-06-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250115586-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF JAK1, JAK3, JAK2 CDK19 167/4885ALK 179/4885CDK2 115/4885
US-12030870-B2 Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof JAK2, JAK1, JAK3 CDK19 103/4885ALK 241/4885CDK2 49/4885
US-20230002362-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF JAK1, JAK3, JAK2 CDK19 167/4885ALK 179/4885CDK2 115/4885
US-20240025882-A1 BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF JAK2, JAK1, JAK3 CDK19 103/4885ALK 241/4885CDK2 49/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.