SCHEMBL22104584

SCHEMBL22104584

Cc1nc(=O)c2cc(CN(C)c3ccc(C(=O)N[C@@H](CCC(=O)NC(C)C)C(=O)O)s3)ccc2[nH]1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.67
DHFR P00374 1/20 0.67
FOLR2 P14207 1/20 0.67
FOLR1 P15328 1/20 0.67
SLC19A1 P41440 1/20 0.67
EHMT2 Q96KQ7 1/20 0.67
SLC46A1 Q96NT5 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Raltitrexed SCHEMBL7439 0.92 TYMS (0.78) TYMSDHFRFOLR2FOLR1SLC19A1
Raltitrexed SCHEMBL29454789 0.92 TYMS (0.78) TYMSDHFRFOLR2FOLR1SLC19A1
Raltitrexed SCHEMBL16766843 0.92 TYMS (0.78) TYMSDHFRFOLR2FOLR1SLC19A1
SCHEMBL3274944 0.92 TYMS (0.70) TYMSDHFRFOLR2FOLR1SLC19A1
SCHEMBL25904644 0.91 TYMS (0.65) TYMSDHFRFOLR2FOLR1SLC19A1
SCHEMBL16366393 0.90 TYMS (0.67) TYMSDHFRFOLR2FOLR1SLC19A1
SCHEMBL22104577 0.89 TYMS (0.85) TYMSDHFRFOLR2FOLR1SLC19A1
SCHEMBL16366259 0.88 TYMS (0.65) TYMSDHFRFOLR2FOLR1SLC19A1
Raltitrexed SCHEMBL28116774 0.88 TYMS (0.72) TYMSDHFRFOLR2FOLR1SLC19A1
Raltitrexed SCHEMBL4954885 0.87 TYMS (0.88) TYMSDHFRFOLR2FOLR1SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020120785-A1 ANTIFOLATE-CARRYING NANOPARTICLES AND THEIR USE IN MEDICINE MIDATECH LTD (GB) 2020-06-18 WO disclosed