SCHEMBL22129205

SCHEMBL22129205

O=C(O)c1cccc2c1C(=O)N(c1ccc(C(F)(F)F)cc1)C2

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 7/20 0.66
TDP1 Q9NUW8 3/20 0.66
KDM4E B2RXH2 1/20 0.66
ESR1 P03372 1/20 0.66
NR4A1 P22736 1/20 0.66
APEX1 P27695 1/20 0.66
PTPN7 P35236 1/20 0.66
RECQL P46063 1/20 0.66
BLM P54132 1/20 0.66
MCL1 Q07820 1/20 0.66
ESR2 Q92731 1/20 0.66
HSD17B10 Q99714 1/20 0.66
PARP1 P09874 6/20 0.52
TP53 P04637 3/20 0.47
HDAC11 Q96DB2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
MAPT P10636 2/20 0.44
HTT P42858 1/20 0.44
ALOX15 P16050 1/20 0.44
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728317 0.85 POLB (0.73) POLBTDP1KDM4EESR1NR4A1
SCHEMBL16907880 0.83 POLB (0.70) POLBTDP1KDM4EESR1NR4A1
SCHEMBL2116520 0.80 POLB (1.00) POLBTDP1KDM4EESR1NR4A1
SCHEMBL835316 0.75 PARP1 (0.79) POLBTDP1KDM4EESR1NR4A1
SCHEMBL22291931 0.74 NPC1 (0.68) KDM4ETP53MAPTHTTNPC1
SCHEMBL6675973 0.72 NPC1 (0.40) POLBTDP1KDM4EESR1NR4A1
SCHEMBL16907926 0.72 POLB (0.56) POLBTDP1KDM4EESR1NR4A1
SCHEMBL16907925 0.71 POLB (0.65) POLBTDP1KDM4EESR1NR4A1
SCHEMBL835757 0.70 PARP1 (0.74) POLBTDP1KDM4EESR1NR4A1
SCHEMBL20096495 0.70 HDAC11 (0.71) HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020124500-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏凯迪恩医药科技有限公司 2020-06-25 WO disclosed