SCHEMBL2213063

SCHEMBL2213063

CC1CCCN(C(=O)c2ccc3cccc(OC4CCN(C(C)C)C4)c3n2)C1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.48
MCHR1 Q99705 7/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
RECQL P46063 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GRM5 P41594 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2209751 0.95 HRH3 (0.53) HRH3MCHR1TP53MAPTRECQL
SCHEMBL2210609 0.90 HRH3 (0.58) HRH3MCHR1NPC1RAB9A
SCHEMBL2208759 0.87 MCHR1 (0.47) HRH3MCHR1
SCHEMBL2214389 0.86 HRH3 (0.52) HRH3MCHR1HCRTR1HCRTR2
SCHEMBL2206388 0.86 HRH3 (0.58) HRH3MCHR1
SCHEMBL2208189 0.85 HRH3 (0.64) HRH3MCHR1
SCHEMBL2208886 0.85 HRH3 (0.61) HRH3MCHR1
SCHEMBL2212774 0.85 HRH3 (0.47) HRH3MCHR1
SCHEMBL2212421 0.84 HRH3 (0.47) HRH3MCHR1
SCHEMBL2211215 0.84 HRH3 (0.57) HRH3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805166-B1 QUINOLINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-07-27 EP claimed