SCHEMBL22149199

SCHEMBL22149199

COc1cc(Nc2ccc3ncc(-c4cnn(C5CCN(C(=O)C6(F)CN(C(=O)/C=C/CN(C)C)C6)CC5)c4)nc3c2)cc(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 20/20 0.49
KDR P35968 19/20 0.49
FGFR4 P22455 18/20 0.48
FGFR1 P11362 18/20 0.48
FGFR2 P21802 16/20 0.48
FLT3 P36888 8/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31655657 1.00 FGFR3 (0.49) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL31655643 0.96 FGFR3 (0.48) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL31655641 0.91 FGFR3 (0.48) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL22149194 0.91 FGFR3 (0.48) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL31655652 0.90 FGFR3 (0.53) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL22149691 0.90 FGFR3 (0.53) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL22149354 0.89 FGFR3 (0.40) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL31655635 0.89 FGFR3 (0.40) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL31655625 0.88 FGFR3 (0.52) FGFR3KDRFGFR4FGFR1FGFR2
SCHEMBL22149123 0.87 FGFR3 (0.41) FGFR3KDRFGFR4FGFR1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020131674-A1 7-((3,5-DIMETHOXYPHENYL)AMINO)QUINOXALINE DERIVATIVES AS FGFR INHIBITORS FOR TREATING CANCER ARRAY BIOPHARMA INC. (US) 2020-06-25 WO disclosed