SCHEMBL22172245

SCHEMBL22172245

Cn1cc2cc(Br)cc(C(F)(F)F)c2n1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
EPRS1 P07814 1/20 0.35
CYP1A2 P05177 1/20 0.32
LRRK2 Q5S007 1/20 0.32
TLR8 Q9NR97 2/20 0.32
LMNA P02545 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NSD2 O96028 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
PDE3B Q13370 2/20 0.30
PDE3A Q14432 2/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31600826 0.79 KDM4E (0.40) CYP1A2LRRK2TLR8KDM4ENSD2
SCHEMBL18081458 0.77 KDM4E (0.33) HTTKDM4ENSD2ALDH1A1MAPT
SCHEMBL17875687 0.77 PRNP (0.42) HTTLMNAKDM4ENSD2ALDH1A1
SCHEMBL3978933 0.75 NQO2 (0.41) HTTLMNAKDM4ENSD2ALDH1A1
SCHEMBL25317472 0.74 TLR8 (0.42) EPRS1TLR8
SCHEMBL31210637 0.74 KDM4E (0.33) KDM4ENSD2ALDH1A1MAPT
SCHEMBL29303414 0.74 NMT1 (0.42) HTTKDM4ENSD2ALDH1A1MAPT
SCHEMBL25227561 0.74 NSD1 (0.42) HTTLMNAKDM4ENSD2ALDH1A1
SCHEMBL31210645 0.74 KDM4E (0.33) KDM4ENSD2ALDH1A1MAPT
SCHEMBL26664175 0.73 KDM4E (0.31) KDM4ENSD2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025111547-A1 2,3-DIHYDROPYROLLOPYRIDINE CARBOXAMIDE COMPOUNDS AND METHODS OF USE THEREOF RGENTA THERAPEUTICS, INC. (US) 2025-05-30 WO disclosed
CN-117769546-A Allosteric ketene inhibitors of phosphoinositide 3-kinase (PI 3K) for the treatment of disease 佩特拉制药公司 2024-03-26 CN disclosed
WO-2020135507-A1 POLYSUBSTITUTED ANILINOPYRIMIDINE DERIVATIVE AND PREPARATION METHOD AND APPLICATION THEREOF 杭州百新生物医药科技有限公司 2020-07-02 WO disclosed