SCHEMBL22200417

SCHEMBL22200417

COc1cc2cc(C(F)(F)CCC(=O)N(O)Cc3ccccc3)sc2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 4/20 0.46
ACHE P22303 11/20 0.43
CLK1 P49759 1/20 0.41
DYRK1A Q13627 1/20 0.41
ALOX5 P09917 2/20 0.40
RXFP1 Q9HBX9 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200400 0.89 CLK1 (0.46) STING1CLK1
SCHEMBL22200395 0.85 STING1 (0.43) STING1ACHE
SCHEMBL22200292 0.85 STING1 (0.46) STING1
SCHEMBL22200618 0.85 TP53 (0.43) CLK1
SCHEMBL22200402 0.84 STING1 (0.42) STING1ACHE
SCHEMBL22200414 0.84 STING1 (0.47) STING1ACHECLK1DYRK1AALOX5
SCHEMBL22200394 0.82 STING1 (0.44) STING1ACHE
SCHEMBL22200401 0.81 STING1 (0.40) STING1ACHE
SCHEMBL23999274 0.81 STING1 (0.45) STING1ACHE
SCHEMBL22200283 0.80 STING1 (0.58) STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3907221-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-11-10 EP disclosed
WO-2020140894-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 中国科学院上海药物研究所 2020-07-09 WO disclosed