SCHEMBL22200834

SCHEMBL22200834

C=CC(=O)Nc1cc2c(Nc3ccc(Oc4cc5nncn5cn4)c(C)c3)c(C#N)cnc2cc1OCC

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.75
ERBB2 P04626 12/20 0.75
STK4 Q13043 5/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20780773 0.88 EGFR (0.80) EGFRERBB2
SCHEMBL30478673 0.88 EGFR (0.80) EGFRERBB2
SCHEMBL22076954 0.88 EGFR (0.63) EGFRERBB2
SCHEMBL30478699 0.88 EGFR (0.63) EGFRERBB2
SCHEMBL22076843 0.88 EGFR (0.62) EGFRERBB2
SCHEMBL22076887 0.87 EGFR (0.59) EGFRERBB2STK4
SCHEMBL20780805 0.86 EGFR (0.64) EGFRERBB2
SCHEMBL30478706 0.86 EGFR (0.82) EGFRERBB2
SCHEMBL20780762 0.86 EGFR (0.82) EGFRERBB2
SCHEMBL22076870 0.84 EGFR (0.62) EGFRERBB2STK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed