SCHEMBL22200864

SCHEMBL22200864

C=CC(=O)Nc1ccc2ncnc(Nc3ccc(Oc4cc5nccn5cn4)c(C)c3)c2c1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.63
ERBB2 P04626 8/20 0.63
FYN P06241 6/20 0.53
SRC P12931 6/20 0.53
BLK P51451 1/20 0.51
BMX P51813 1/20 0.51
JAK3 P52333 1/20 0.51
BTK Q06187 1/20 0.51
ERBB4 Q15303 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12888131 0.89 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL20605393 0.89 EGFR (0.78) EGFRERBB2FYNSRC
SCHEMBL24168145 0.87 EGFR (0.57) EGFRERBB2ERBB4
SCHEMBL20780826 0.87 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL20780822 0.87 EGFR (0.59) EGFRERBB2FYNSRCBLK
SCHEMBL22076917 0.86 EGFR (0.60) EGFRERBB2
SCHEMBL20780780 0.86 ERBB2 (0.56) EGFRERBB2
SCHEMBL20780779 0.84 EGFR (0.83) EGFRERBB2
SCHEMBL29025879 0.84 EGFR (0.83) EGFRERBB2
SCHEMBL30478678 0.84 EGFR (0.83) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677583-A1 NITROGENOUS HETEROCYCLIC COMPOUND, PREPARATION METHOD, INTERMEDIATE, COMPOSITION, AND APPLICATION Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2020-07-08 EP disclosed