SCHEMBL22202089

SCHEMBL22202089

COC1=CC=C(Nc2ncc(I)cn2)CC1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
AURKA O14965 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10183405 0.68
SCHEMBL22191045 0.67 HDAC3 (0.59) CDK5CDK5R1AURKASYK
SCHEMBL13839056 0.66 CA1 (0.35)
SCHEMBL12962757 0.63
SCHEMBL19062182 0.62 KMT2A (0.45)
SCHEMBL22191522 0.61 LRRK2 (0.56) AURKA
SCHEMBL22191547 0.59 SYK (0.60) CDK5CDK5R1AURKASYK
SCHEMBL22299742 0.58 LRRK2 (0.47)
SCHEMBL15729997 0.58
SCHEMBL737749 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020142486-A1 KINASE INHIBITOR COMPOUNDS AND COMPOSITIONS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2020-07-09 WO disclosed