SCHEMBL22216504

SCHEMBL22216504

CC(C)(C)Cn1cnc2c(N)nc(Cl)nc21

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.61
PI4K2B Q8TCG2 1/20 0.61
PI4K2A Q9BTU6 1/20 0.61
PI4KB Q9UBF8 1/20 0.61
CDK1 P06493 2/20 0.58
PDE8A O60658 10/20 0.53
CCNB1 P14635 1/20 0.49
CCNE1 P24864 1/20 0.49
CDK2 P24941 1/20 0.49
ADORA3 P0DMS8 2/20 0.43
CFTR P13569 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
YTHDC1 Q96MU7 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16134183 0.84 CCNE1 (0.69) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL179425 0.83 PI4KA (0.63) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL3440998 0.83 CDK1 (0.71) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL23619320 0.81 CDK1 (0.60) CDK1PDE8ACCNB1CCNE1CDK2
SCHEMBL3441081 0.80 CDK1 (0.64) CDK1PDE8ACCNB1CCNE1CDK2
SCHEMBL6884460 0.79 HSP90AB1 (0.55) PI4KAPI4K2BPI4K2API4KB
SCHEMBL24026363 0.79 CDK1 (0.58) CDK1PDE8ACCNB1CCNE1CDK2
SCHEMBL3441119 0.79 CDK1 (0.58) CDK1PDE8ACCNB1CCNE1CDK2
SCHEMBL179439 0.78 PI4KA (0.57) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL14024978 0.78 ADORA2A (0.62) CDK1PDE8ACCNB1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11034715-B2 Ectonucleotidase inhibitors and methods of use thereof CALITHERA BIOSCIENCES, INC. (US) 2021-06-15 US disclosed
US-20200223882-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2020-07-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200223882-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof NT5E, ENTPD5, NT5C2 PI4KA 3541/4885PI4K2B 4005/4885PI4K2A 3818/4885
US-11034715-B2 Ectonucleotidase inhibitors and methods of use thereof NT5E, ENTPD5, NT5C2 PI4KA 3541/4885PI4K2B 4005/4885PI4K2A 3818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.