SCHEMBL22230705

SCHEMBL22230705

COCOc1ccc(Br)nc1F

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 1/20 0.33
KCNN4 O15554 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
MAPT P10636 1/20 0.30
XDH P47989 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30785978 1.00 S1PR4 (0.33) S1PR4KCNN4ADORA2AADORA1MAPT
SCHEMBL16238204 0.81 S1PR4 (0.33) S1PR4KCNN4XDH
SCHEMBL16742675 0.80 S1PR4 (0.34) S1PR4ADORA2AADORA1MAPTXDH
SCHEMBL30082515 0.80 S1PR4 (0.34) S1PR4ADORA2AADORA1MAPTXDH
SCHEMBL5455137 0.79 NQO2 (0.39) MAPT
SCHEMBL31556399 0.79 NQO2 (0.39) MAPT
SCHEMBL2370651 0.79 CLCN2 (0.35) S1PR4KCNN4XDH
SCHEMBL28566471 0.79 KMT2A (0.33) S1PR4ADORA2AADORA1MAPTXDH
SCHEMBL24992633 0.77 S1PR4 (0.33) S1PR4ADORA2AADORA1MAPTXDH
SCHEMBL30865588 0.77 S1PR4 (0.33) S1PR4ADORA2AADORA1MAPTXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112771027-B Lysophosphatidic acid receptor antagonists and process for preparing the same 武汉朗来科技发展有限公司 2024-03-05 CN disclosed
CN-112771027-A Lysophosphatidic acid receptor antagonists and process for their preparation 武汉朗来科技发展有限公司 2021-05-07 CN disclosed
WO-2020147739-A1 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND PREPARATION METHOD THEREFOR 武汉朗来科技发展有限公司 2020-07-23 WO disclosed