SCHEMBL22237459

SCHEMBL22237459

COc1ccc(CN2CCOC(Cc3cccc(Cc4ccccc4)c3)C2=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.49
DRD4 P21917 2/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
SIGMAR1 Q99720 2/20 0.43
LTA4H P09960 1/20 0.43
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.39
OPRK1 P41145 1/20 0.39
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
CLPP Q16740 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20832666 0.90 TACR1 (0.46) TACR1DRD4DRD2DRD3SIGMAR1
SCHEMBL22623154 0.88 MAPT (0.51) TACR1DRD4DRD2DRD3SIGMAR1
SCHEMBL22227848 0.85 TACR1 (0.44) TACR1DRD4DRD2DRD3SIGMAR1
SCHEMBL14154859 0.81 DRD4 (0.51) TACR1DRD4MEN1KMT2AGAA
SCHEMBL1553056 0.80 TACR1 (0.56) TACR1MEN1KMT2ACLPP
SCHEMBL1551999 0.78 TACR1 (0.56) TACR1SIGMAR1MEN1KMT2ACLPP
SCHEMBL5968243 0.78 TACR1 (0.56) TACR1DRD2DRD3SIGMAR1
SCHEMBL5667214 0.78 TACR1 (0.56) TACR1DRD2DRD3SIGMAR1
SCHEMBL1553263 0.77 TACR1 (0.53) TACR1DRD4
SCHEMBL6493798 0.76 TACR1 (0.43) TACR1DRD4DRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3682881-A1 COMPOUND HAVING CYCLIC STRUCTURE DAIICHI SANKYO COMPANY, LIMITED (JP) 2020-07-22 EP disclosed