SCHEMBL2226121

SCHEMBL2226121

O=CCc1cc2ccc(Br)cc2cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.41
CYP2A6 P11509 2/20 0.38
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ERN1 O75460 1/20 0.35
TLR2 O60603 1/20 0.34
GSK3A P49840 1/20 0.33
CDK9 P50750 1/20 0.33
CDK5 Q00535 1/20 0.33
TAOK1 Q7L7X3 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
THRB P10828 1/20 0.33
NOS1 P29475 2/20 0.33
METAP2 P50579 2/20 0.33
CYP1A2 P05177 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23174730 0.79 ATM (0.47) CYP2A6KDM4EMAPTCYP1A2L3MBTL1
SCHEMBL2226466 0.77 ABL1 (0.44) ABL1CYP2A6KDM4EMEN1ALDH1A1
SCHEMBL10272932 0.77 CYP2A6 (0.42) ABL1CYP2A6KDM4EMEN1ALDH1A1
SCHEMBL30718639 0.77 ABL1 (0.44) ABL1CYP2A6KDM4EMEN1ALDH1A1
SCHEMBL28300308 0.77 ABL1 (0.37) ABL1CYP2A6KDM4EMEN1ALDH1A1
SCHEMBL1641540 0.75 ABL1 (0.42) ABL1CYP2A6KDM4EMEN1ALDH1A1
SCHEMBL266084 0.75 BACE1 (0.49) CYP2A6KDM4EMEN1ALDH1A1MAPT
SCHEMBL525153 0.74 CYP2A6 (0.46) CYP2A6KDM4EMEN1ALDH1A1MAPT
SCHEMBL622260 0.74 GBA1 (0.41) KDM4EALDH1A1MAPTKMT2A
SCHEMBL29600434 0.74 GBA1 (0.41) KDM4EALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091446-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-07-28 WO disclosed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed