SCHEMBL2226141

SCHEMBL2226141

[CH2]Cc1ccc(-c2cnc(N)c(C(=O)Nc3cccnc3)n2)cc1

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.72
CCNE2 O96020 10/20 0.72
CCNE1 P24864 10/20 0.72
CDK2 P24941 10/20 0.72
ATR Q13535 9/20 0.69
CYP3A4 P08684 1/20 0.69
PRKDC P78527 2/20 0.64
GSK3A P49840 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230199 0.93 GSK3B (0.68) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL9907070 0.91 ATR (0.80) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL2226149 0.90 GSK3B (0.71) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL411857 0.89 GSK3B (0.70) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6616616 0.88 ATR (0.78) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL9907069 0.88 GSK3B (0.70) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL413176 0.88 GSK3B (0.67) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6615544 0.88 ATR (0.88) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6620408 0.87 ATR (0.79) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6619968 0.87 ATR (0.81) GSK3BCCNE2CCNE1CDK2ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011089416-A1 PYRAZINE DERIVATIVES ASTRAZENECA AB (SE) 2011-07-28 WO disclosed