SCHEMBL2226174

SCHEMBL2226174

CCCOc1ccc(C=CC(N)=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.63
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
CYP1A1 P04798 1/20 0.58
CYP1B1 Q16678 1/20 0.58
SAE1 Q9UBE0 1/20 0.55
UBA2 Q9UBT2 1/20 0.55
PTGS1 P23219 1/20 0.54
PTGS2 P35354 1/20 0.54
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
LMNA P02545 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
GAA P10253 1/20 0.49
MAPT P10636 2/20 0.49
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49
TUBA4A P68366 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9716959 0.89 ABCG2 (0.59) ABCG2NPC1RAB9ASAE1UBA2
SCHEMBL2225311 0.87 NPC1 (0.63) ABCG2NPC1RAB9AKMT2AMEN1
SCHEMBL8149314 0.87 NPC1 (0.63) ABCG2NPC1RAB9AKMT2AMEN1
SCHEMBL4933565 0.85 ABCG2 (0.65) ABCG2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL417824 0.85 ABCG2 (0.65) ABCG2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL417823 0.85 ABCG2 (0.65) ABCG2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL4933573 0.85 ABCG2 (0.65) ABCG2NPC1RAB9ACYP1A1CYP1B1
Hydrochloric Acid SCHEMBL7054655 0.84 ABCG2 (0.63) ABCG2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL7054652 0.84 ABCG2 (0.63) ABCG2NPC1RAB9ACYP1A1CYP1B1
SCHEMBL7054651 0.84 ABCG2 (0.63) ABCG2NPC1RAB9ACYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083413-A1 PIPERAZINES AS ANTIMALARIAL AGENTS ACTELION PHARMACEUTICALS LTD (CH) 2011-07-14 WO disclosed