SCHEMBL22266262

SCHEMBL22266262

OCCOCCOCc1ccon1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
APP P05067 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
S1PR1 P21453 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22266264 0.96 TSHR (0.33) MEN1KMT2ATSHRMAPK1
SCHEMBL22266258 0.93 TSHR (0.34) MEN1KMT2ATSHRMAPK1
SCHEMBL22266268 0.90 CYP1A2 (0.30)
SCHEMBL22266282 0.86 MEN1 (0.39) MEN1KMT2ATSHRMAPK1APP
SCHEMBL22266320 0.86 CYP1A2 (0.32)
SCHEMBL22266278 0.84 HDAC3 (0.33)
SCHEMBL20235114 0.84 MAPK1 (0.37) MEN1KMT2ATSHRMAPK1
SCHEMBL22266313 0.83 HDAC3 (0.33)
SCHEMBL22266274 0.83 HDAC3 (0.33)
SCHEMBL24761891 0.82 CYP1A2 (0.32) APPL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10723717-B2 Compounds and methods for the targeted degradation of rapidly accelerated fibrosarcoma polypeptides ARVINAS OPERATIONS, INC. (US) 2020-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10723717-B2 Compounds and methods for the targeted degradation of rapidly accelerated fibrosarcoma polypeptides CRBN, ARAF, VHL MEN1 2317/4885KMT2A 1975/4885TSHR 2304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.