SCHEMBL22280306

SCHEMBL22280306

COc1ccc(-c2noc(C3CNC3)n2)cc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.53
TLR9 Q9NR96 4/20 0.48
TLR8 Q9NR97 4/20 0.48
TLR7 Q9NYK1 4/20 0.48
NPSR1 Q6W5P4 1/20 0.45
SPHK2 Q9NRA0 2/20 0.43
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
S1PR5 Q9H228 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22280452 0.90 HTR2A (0.53) S1PR1TLR9TLR8TLR7SPHK2
SCHEMBL22280635 0.85 S1PR1 (0.54) S1PR1TLR9TLR8TLR7NR1H4
Hydrochloric Acid SCHEMBL22265746 0.83 SPHK2 (0.62) S1PR1TLR9TLR8TLR7SPHK2
Hydrochloric Acid SCHEMBL22265618 0.83 SPHK2 (0.62) S1PR1TLR9TLR8TLR7SPHK2
SCHEMBL22280463 0.81 SPHK2 (0.62) S1PR1SPHK2
Hydrochloric Acid SCHEMBL29523175 0.81 SPHK2 (0.62) S1PR1SPHK2
SCHEMBL22280631 0.80 S1PR1 (0.46) S1PR1SPHK2L3MBTL1
Hydrochloric Acid SCHEMBL29523923 0.79 SPHK2 (0.47) S1PR1SPHK2L3MBTL1
SCHEMBL25433735 0.76 MAPT (0.54) S1PR1NPSR1NR1H4MEN1CYP3A4
Hydrochloric Acid SCHEMBL22265421 0.76 SPHK2 (0.46) TLR9TLR8TLR7SPHK2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020154431-A1 INHIBITORS OF SPINSTER HOMOLOG 2 (SPNS2) FOR USE IN THERAPY LYNCH KEVIN R (US) 2020-07-30 WO disclosed