SCHEMBL22282186

SCHEMBL22282186

Clc1nc(N2CC3(CCCCC3)C2)c2cn[nH]c2n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.39
PDE2A O00408 1/20 0.38
PLK4 O00444 1/20 0.35
PAK4 O96013 1/20 0.35
RPS6KB1 P23443 2/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
AKT2 P31751 2/20 0.32
SGK1 O00141 7/20 0.32
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31106994 0.84 SGK1 (0.38) PDE2APLK4PAK4RPS6KB1HTR2A
SCHEMBL24672317 0.74 AKT2 (0.38) PDE2APLK4PAK4AKT2SGK1
SCHEMBL3984786 0.73 PIK3CA (0.49) RPS6KB1HTR2AHTR2CAKT2SGK1
SCHEMBL31107020 0.70 SGK1 (0.38) PDE2APLK4PAK4AKT2SGK1
SCHEMBL55757 0.70 MTOR (0.40) PDE2APLK4PAK4AKT2SGK1
SCHEMBL24955620 0.70 SGK1 (0.38) PDE2APLK4PAK4AKT2SGK1
SCHEMBL53863 0.65 PLK4 (0.47) PDE2APLK4PAK4ALDH1A1SMN1; SMN2
SCHEMBL2266999 0.62 PLK4 (0.45) PDE2APLK4PAK4ALDH1A1SMN1; SMN2
SCHEMBL560806 0.62 RET (0.52) PDE2APLK4PAK4HTR2AHTR2C
SCHEMBL61883 0.62 PLK4 (0.53) PDE2APLK4PAK4HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020151707-A1 NOVEL SMALL MOLECULE CD73 INHIBITOR, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 江苏恒瑞医药股份有限公司 2020-07-30 WO disclosed