SCHEMBL22296233

SCHEMBL22296233

CC(C)c1ccc(N2CCC(O)C(C)(C)C2)cn1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 3/20 0.36
HRH3 Q9Y5N1 5/20 0.35
EGFR P00533 4/20 0.35
BTK Q06187 1/20 0.35
PANK3 Q9H999 1/20 0.33
ESR1 P03372 1/20 0.33
ACACB O00763 1/20 0.33
LCAT P04180 2/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23866054 0.88 CCR6 (0.34) CCR6HRH3ESR1ACACBNR1H2
SCHEMBL22296208 0.83 CHRM4 (0.39) EGFRBTK
SCHEMBL17660305 0.81 MAPT (0.46) CCR6HRH3
SCHEMBL24746187 0.81 PIK3CA (0.37) HRH3EGFRBTK
SCHEMBL24747235 0.81 PIK3CA (0.37) HRH3EGFRBTK
SCHEMBL23865949 0.81 EGFR (0.36) HRH3EGFRBTKLCAT
SCHEMBL17055343 0.81 PIK3CA (0.37) HRH3EGFRBTK
SCHEMBL23108883 0.80 CCR6 (0.43) CCR6
SCHEMBL23103745 0.80 CCR6 (0.43) CCR6
SCHEMBL23114413 0.80 CCR6 (0.43) CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3689871-B1 4,6,7-TRISUBSTITUTED 1,2-DIHYDROPYRROL[3,4-C]PYRIDIN/PYRIMIDIN-3-ONE DERIVATIVE AND USE SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (CN) 2021-09-29 EP disclosed
EP-3689871-A1 4,6,7-TRISUBSTITUTED 1,2-DIHYDROPYRROL[3,4-C]PYRIDIN/PYRIMIDIN-3-ONE DERIVATIVE AND USE Shanghai Haiyan Pharmaceutical Technology Co., Ltd. (CN) 2020-08-05 EP disclosed