SCHEMBL22297643

SCHEMBL22297643

C/C=C\C=C/C(C)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RCE1 Q9Y256 1/20 0.41
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.36
SLC1A3 P43003 2/20 0.36
SLC1A2 P43004 2/20 0.36
SLC1A1 P43005 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
IDO1 P14902 1/20 0.35
AGXT P21549 1/20 0.34
ALDH1A1 P00352 2/20 0.34
HTT P42858 3/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31453504 0.87 RCE1 (0.44) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL5139238 0.87 RCE1 (0.44) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL7228724 0.80 TSHR (0.44) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL7157545 0.79 RCE1 (0.43) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL20034084 0.78 RCE1 (0.35) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL3127875 0.75 HCAR2 (0.51) RCE1TSHRSLC1A3SLC1A2SLC1A1
SCHEMBL3127891 0.75 HCAR2 (0.51) RCE1TSHRSLC1A3SLC1A2SLC1A1
SCHEMBL6172748 0.74 SLC1A3 (0.47) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL9250351 0.74 RCE1 (0.45) RCE1TSHRMAPTSLC1A3SLC1A2
SCHEMBL6239311 0.74 SLC1A3 (0.47) RCE1TSHRMAPTSLC1A3SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3689868-A1 TETRAHYDRONAPHTHALENE AND TETRAHYDROISOQUINOLINE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS Arvinas Operations, Inc. (US) 2020-08-05 EP disclosed