SCHEMBL22323738

SCHEMBL22323738

C=C1C(OCc2ccccc2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 2/20 0.46
STS P08842 1/20 0.44
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
GPR119 Q8TDV5 2/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
LMNA P02545 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
KDM1A O60341 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
GAA P10253 1/20 0.40
THRB P10828 1/20 0.40
YAP1 P46937 1/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27579467 0.79 KLK7 (0.46) KLK7STSGPR119JAK2JAK1
SCHEMBL22324617 0.78 ABCB1 (0.42) KLK7STSGPR119JAK2JAK1
SCHEMBL21996514 0.78 ABCB1 (0.42) KLK7STSGPR119JAK2JAK1
SCHEMBL3249107 0.76 STS (0.58) STSGPR119JAK2JAK1LMNA
SCHEMBL21996403 0.76 KDM1A (0.39) GPR119KDM4EKDM1ASMN1; SMN2THRB
SCHEMBL15720471 0.76 STS (0.47) KLK7STSDDB1CRBNGPR119
SCHEMBL24535177 0.74 STS (0.48) KLK7STSDDB1CRBNGPR119
SCHEMBL22355152 0.74 TMEM97 (0.43) KLK7STSGPR119LMNAKDM4E
SCHEMBL942191 0.74 JAK2 (0.55) KLK7STSGPR119JAK2JAK1
SCHEMBL20503925 0.74 JAK2 (0.55) KLK7STSGPR119JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109232350-A A method of preparing N-Boc-3- pyrrolidine formaldehyde 辽宁东科药业有限公司 2019-01-18 CN claimed
WO-2020113077-A9 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-08-13 WO disclosed
CN-109232350-A A method of preparing N-Boc-3- pyrrolidine formaldehyde 辽宁东科药业有限公司 2019-01-18 CN disclosed
CN-109232350-A A method of preparing N-Boc-3- pyrrolidine formaldehyde 辽宁东科药业有限公司 2019-01-18 CN disclosed