SCHEMBL22325529

SCHEMBL22325529

O=C(O)c1cccc(COc2ccc(-n3cncn3)nc2)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 15/20 0.56
TP53 P04637 2/20 0.52
PKM P14618 2/20 0.52
NFKB1 P19838 2/20 0.52
NFKB2 Q00653 2/20 0.52
RELA Q04206 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
RAB9A P51151 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
CYP4F2 P78329 2/20 0.52
CYP4A11 Q02928 2/20 0.52
ALKBH1 Q13686 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22335795 0.89 CYP4F2 (0.55) MRGPRX4SMN1; SMN2CYP4F2CYP4A11ALKBH1
SCHEMBL20590806 0.84 NPC1 (0.54) TP53NFKB1NFKB2RELASMN1; SMN2
SCHEMBL22325491 0.82 CYP4F2 (0.61) MRGPRX4SMN1; SMN2RAB9ACYP4F2CYP4A11
SCHEMBL22968107 0.80 CYP4F2 (0.53) CYP4F2CYP4A11
SCHEMBL22335800 0.76 CYP4F2 (0.53) CYP4F2CYP4A11
SCHEMBL15167297 0.75 EGLN1 (0.74) ALKBH1
SCHEMBL22335796 0.74 MAPT (0.51) SMN1; SMN2CYP4F2CYP4A11
SCHEMBL600130 0.74 MAPT (0.64) SMN1; SMN2
SCHEMBL18906070 0.74 MRGPRX4 (0.67) MRGPRX4TP53PKMNFKB1NFKB2
SCHEMBL22480878 0.72 MRGPRX4 (1.00) MRGPRX4TP53PKMNFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020162612-A1 PYRIDINE COMPOUND SUBSTITUTED BY HETEROARYL 大正製薬株式会社 2020-08-13 WO disclosed