SCHEMBL223290

SCHEMBL223290

C[C@@H]1CC2=CC(=O)CC[C@@H]2[C@H]2CC[C@]3(C)[C@@H](O)CC[C@H]3[C@@H]21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 1.00
SHBG P04278 7/20 0.69
SERPINA6 P08185 2/20 0.69
SLC22A1 O15245 1/20 0.69
ALDH1A1 P00352 1/20 0.69
THRB P10828 1/20 0.69
PGR P06401 5/20 0.55
NR3C2 P08235 2/20 0.55
CYP19A1 P11511 1/20 0.50
PDK1 Q15118 1/20 0.48
PDK2 Q15119 1/20 0.48
PDK3 Q15120 1/20 0.48
PDK4 Q16654 1/20 0.48
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25863609 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL1255845 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL29880093 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL5188310 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL24102494 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL14342101 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL24103284 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL5026430 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL24103286 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1
SCHEMBL199806 1.00 AR (1.00) ARSHBGSERPINA6SLC22A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 999 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3441089-B1 TREATMENT METHODS USING ADENOVIRUS VASCULAR BIOGENICS LTD (IL) 2022-12-14 EP claimed
EP-3191114-B1 OCCIDIOFUNGIN FORMULATIONS AND USES THEREOF UNIV MISSISSIPPI STATE (US) 2021-03-03 EP claimed
EP-2908865-B1 ADENOVIRUS EXPRESSING A FAS-CHIMERA AND USE THEREOF IN CANCER TREATMENT METHODS VASCULAR BIOGENICS LTD (IL) 2018-10-03 EP claimed
EP-2923703-B1 TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS NANTBIO INC (US) 2018-09-19 EP claimed
EP-3368081-A1 TREATMENT OF CANCER WITH COMBINATIONS OF RXR AGONISTS AND THYROID HORMONES IO Therapeutics, Inc. (US) 2018-09-05 EP claimed
EP-3124481-B1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS INC (US) 2018-03-28 EP claimed
US-20170348321-A1 Wafer Comprising Steroid Hormones LTS LOHMANN THERAPIE-SYSTEME AG (DE) 2017-12-07 US claimed
US-9763960-B2 Wafer comprising steroid hormones LTS LOHMANN THERAPLE-SYSTEME AG (DE) 2017-09-19 US claimed
WO-2017075612-A1 TREATMENT OF CANCER WITH COMBINATIONS OF RXR AGONISTS AND THYROID HORMONES Io Therapeutics, Inc. (US) 2017-05-04 WO claimed
US-9364488-B2 Myelin regeneration with androgens THE POPULATION COUNCIL, INC. (US) 2016-06-14 US claimed
WO-2003079961-A2 METHOD FOR PRODUCING 7$G(A)-METHYL STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-02 WO claimed
WO-2003068314-A1 PULMONARY ADMINISTRATION OF 6-ALPHA-ALKYLATED TESTOSTERONE DERIVATIVES FOR ANDROGEN REPLACEMENT THERAPY PANTARHEI BIOSCIENCE B.V. (NL) 2003-08-21 WO claimed
US-20030096739-A1 Nuclear receptor-mediated introduction of a PNA into cell nuclei POPULATION COUNCIL, INC., THE 2003-05-22 US claimed
WO-2002083186-A1 NUCLEAR RECEPTOR-MEDIATED INTRODUCTION OF A PNA INTO CELL NUCLEI THE POPULATION COUNCIL, INC. (US) 2002-10-24 WO claimed
EP-0970704-B1 Silicone core long term androgen delivery implant POPULATION COUNCIL INC (US) 2002-09-11 EP claimed
US-20020012694-A1 TRANSDERMAL ADMINISTRATION OF MENT POPULATION COUNCIL, INC., THE, A CORP. OF NY 2002-01-31 US claimed
US-6117441-A Silicone core long term androgen delivery implant THE POPULATION COUNCIL, INC. (US) 2000-09-12 US claimed
EP-0941039-A1 TRANSDERMAL ADMINISTRATION OF MENT THE POPULATION COUNCIL, INC. (US) 1999-09-15 EP claimed
WO-1999013812-A1 TRANSDERMAL ADMINISTRATION OF MENT THE POPULATION COUNCIL, INC. (US) 1999-03-25 WO claimed
US-5342834-A Administering testosterone derivatives THE POPULATION COUNCIL, INC. (US) 1994-08-30 US claimed