SCHEMBL22335209

SCHEMBL22335209

N=C(N)c1cc(C(=O)O)ccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.50
LMNA P02545 1/20 0.47
KDM4E B2RXH2 10/20 0.47
KMT2A Q03164 2/20 0.47
GFER P55789 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
MAPT P10636 5/20 0.46
THRB P10828 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
POLB P06746 3/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
PKM P14618 1/20 0.46
APEX1 P27695 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
MCL1 Q07820 1/20 0.46
GLA P06280 2/20 0.44
KEAP1 Q14145 1/20 0.44
ALDH1A1 P00352 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22335212 0.85 CDC25B (0.46) CDC25BLMNAKDM4EGFERMAPT
SCHEMBL13688528 0.84 IKBKB (0.56) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL5248866 0.84 KDM4E (0.48) CDC25BLMNAKDM4EMAPTTDP1
SCHEMBL265109 0.84 KDM4E (0.65) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL29593435 0.84 KDM4E (0.65) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL13522728 0.83 CDC25B (0.49) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL11542659 0.82 KDM4E (0.63) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL18829004 0.80 CDC25B (0.46) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL5707615 0.78 CDC25B (0.52) CDC25BLMNAKDM4EKMT2AGFER
SCHEMBL18828998 0.76 CDC25B (0.42) CDC25BLMNAKDM4EKMT2AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134408-B1 FACTOR XIa INHIBITORS MERCK SHARP & DOHME (US) 2020-08-12 EP disclosed