SCHEMBL22345162

SCHEMBL22345162

O=C(O)c1cnc(N2CC(CO)(CO)C2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.53
P4HA1 P13674 2/20 0.39
P4HTM Q9NXG6 2/20 0.39
OGA O60502 1/20 0.37
RBP4 P02753 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HCAR3 P49019 6/20 0.35
HCAR2 Q8TDS4 1/20 0.34
MIF P14174 1/20 0.34
HDAC3 O15379 4/20 0.33
HDAC1 Q13547 4/20 0.33
HDAC2 Q92769 4/20 0.33
HDAC8 Q9BY41 4/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22345180 0.84 POLB (0.50) POLBP4HA1P4HTMOGARBP4
SCHEMBL22345184 0.78 POLB (0.44) POLBOGAKDM4EALDH1A1ALOX15
SCHEMBL16824215 0.75 POLB (0.59) POLBP4HA1P4HTMOGARBP4
SCHEMBL34472207 0.73 POLB (0.53) POLBOGARBP4HDAC3HDAC1
SCHEMBL184998 0.73 POLB (0.71) POLBP4HA1P4HTMOGARBP4
SCHEMBL28590337 0.72 POLB (0.55) POLBOGARBP4KDM4EALDH1A1
SCHEMBL186135 0.72 POLB (0.69) POLBOGARBP4KDM4EALDH1A1
SCHEMBL8208254 0.71 POLB (0.58) POLBOGAKDM4EHDAC3HDAC1
SCHEMBL16827289 0.70 POLB (0.61) POLBOGARBP4KDM4EALDH1A1
SCHEMBL23157959 0.69 POLB (0.65) POLBP4HA1P4HTMOGARBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed